Kinetic Assays

“We are experts in the development and application of kinetic assays to measure the association and dissociation rates of unlabelled¬†ligands.”

We have extensive experience of utilizing competition association assays in both radioligand and time-resolved fluorescence resonance energy transfer (TR-FRET) formats.

Assays are medium throughput (384 well), capable of performing fragment screening. We have experience on a range of target classes, including GPCRs, enzymes and protein-protein interactions.

Press Release: Cisbio and Excellerate Bioscience partner on ligand kinetic binding services.

Also watch a webinar from Prof Charlton in collaboration with BMG Labtech and Cisbio and on why and how to measure receptor kinetics in drug discovery programs: